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Eletriptan hydrobromide
CAS No. 177834-92-3
Eletriptan hydrobromide( UK 116044 hydrobromide )
Catalog No. M12677 CAS No. 177834-92-3
Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 30 | In Stock |
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| 5MG | 47 | In Stock |
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| 10MG | 58 | In Stock |
|
| 25MG | 122 | In Stock |
|
| 50MG | 222 | In Stock |
|
| 100MG | 405 | In Stock |
|
| 200MG | 527 | In Stock |
|
| 500MG | 843 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEletriptan hydrobromide
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NoteResearch use only, not for human use.
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Brief DescriptionEletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.
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DescriptionEletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist; significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease; displays antimigraine activity.Migrainev Approved.
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In Vitro——
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In Vivo——
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SynonymsUK 116044 hydrobromide
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PathwayGPCR/G Protein
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Target5-HT Receptor
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Recptor5-HT1B|5-HT1D
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Research AreaNeurological Disease
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IndicationMigraine
Chemical Information
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CAS Number177834-92-3
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Formula Weight463.43
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Molecular FormulaC22H26N2O2S.HBr
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Purity>98% (HPLC)
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SolubilityDMSO: 46.3 mg/mL (100 mM) （ < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESCN1CCC[C@@H]1CC2=CNC3=C2C=C(C=C3)CCS(=O)(=O)C4=CC=CC=C4.Br
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Chemical Name3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.
2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.
3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.
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