Eletriptan hydrobromide

CAS No. 177834-92-3

Eletriptan hydrobromide ( UK 116044 hydrobromide )

Catalog No. M12677 CAS No. 177834-92-3

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 30 In Stock
5MG 47 In Stock
10MG 58 In Stock
25MG 122 In Stock
50MG 222 In Stock
100MG 405 In Stock
200MG 527 In Stock
500MG 843 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Eletriptan hydrobromide
  • Note
    Research use only, not for human use.
  • Brief Description
    Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist.
  • Description
    Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist; significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease; displays antimigraine activity.Migrainev Approved
  • Synonyms
    UK 116044 hydrobromide
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT1B;5-HT1D
  • Research Area
    Neurological Disease
  • Indication
    Migraine

Chemical Information

  • CAS Number
    177834-92-3
  • Formula Weight
    463.43
  • Molecular Formula
    C22H26N2O2S.HBr
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 46.3 mg/mL (100 mM) ( < 1 mg/ml refers to the product slightly soluble or insoluble )
  • SMILES
    CN1CCC[C@@H]1CC2=CNC3=C2C=C(C=C3)CCS(=O)(=O)C4=CC=CC=C4.Br
  • Chemical Name
    3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.
2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.
3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.
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